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Palbociclib-propargyl是一种PROTAC靶蛋白CDK6的配体,可通过PEGlinker与CRBN配体结合,组成PROTACCP-10。CP-10可降解CDK6,DC50值为2.1nM。
Palbociclib-propargyl is a ligand for target protein CDK6 for PROTAC, and binds to CRBN ligand via a PEG linker to make a PROTAC CP-10. CP-10 shows a DC50 of 2.1 nM for CDK6[1].
[1]. Su S, et al. Potent and Preferential Degradation of CDK6 via Proteolysis Targeting Chimera Degraders. J Med Chem. 2019 Aug 22;62(16):7575-7582.
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