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  • Stafia-1
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Stafia-1

Stafia-1 is the first STAT5a inhibitor that inhibits STAT5a (IC50=22.2?μM, Ki=10.9?μM) with at least 9‐fold selectivity over STAT5b and higher selectivity against other STAT family members.

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¥2437-20300
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1950-16240
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  • 货号: ajcx33962
  • CAS: 2582757-90-0
  • 别名:
  • 分子式: C24H27O10P
  • 分子量: 506.44
  • 纯度: >98%
  • 溶解度: DMSO : 250 mg/mL (493.64 mM; Need ultrasonic)
  • 储存: Store at -20°C
  • 库存: 现货

Background

Stafia-1 is the first STAT5a inhibitor that inhibits STAT5a (IC50=22.2?μM, Ki=10.9?μM) with at least 9‐fold selectivity over STAT5b and higher selectivity against other STAT family members.


[1] Natarajan K, et al. Chemistry. 2020 Jan 2;26(1):148-154.

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