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  • Tolebrutinib
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Tolebrutinib

Tolebrutinib (SAR442168, PRN2246, BTKi'168, BTKi('168)) is an oral, CNS-penetrant, irreversible inhibitor of Bruton's tyrosine kinase (BTK) with IC50s of 0.4 nM and 0.7 nM in Ramos B cells and in HMC microglia cells, respectively.

原价
¥3775-26712
价格
3020-21370
Tolebrutinib的二维码

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  • 库存: 现货
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  • 货号: ajcx35276
  • CAS: 1971920-73-6
  • 别名: SAR442168; PRN2246
  • 分子式: C26H25N5O3
  • 分子量: 455.51
  • 纯度: >98%
  • 溶解度: DMSO : 100 mg/mL (219.53 mM; Need ultrasonic)
  • 储存: Store at -20°C
  • 库存: 现货

Background

Tolebrutinib (SAR442168, PRN2246, BTKi'168, BTKi('168)) is an oral, CNS-penetrant, irreversible inhibitor of Bruton's tyrosine kinase (BTK) with IC50s of 0.4 nM and 0.7 nM in Ramos B cells and in HMC microglia cells, respectively.


[1] Francesco MR, et, al. Multiple Sclerosis Journal. 2017;Poster Session 2:P989. [2] Daniel S Reich, et, al. Lancet Neurol. 2021 Sep;20(9):729-738.

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