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  • CAY10573
CAY10573的可视化放大

CAY10573

A PPAR pan-agonist

原价
¥712-10062
价格
570-8050
CAY10573的二维码

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  • 货号: ajci70590
  • CAS: 853652-40-1
  • 别名:
  • 分子式: C33H31NO5
  • 分子量: 521.6
  • 纯度: >98%
  • 溶解度: DMF: 0.3 mg/ml,DMSO: 0.5 mg/ml
  • 储存: Store at -20°C
  • 库存: 现货

Background

The peroxisome proliferator-activated receptors (PPARs) are lipid-activated transcription factors often used as drug targets for the treatment of metabolic disorders. CAY10573 is a PPAR agonist that displays potent binding at PPARα, γ, and δ with IC50 values of 113, 50, and 223 nM, respectively. It potently transactivates PPARα, γ, and δ with EC50 values of 8, 70, and 500 nM, respectively. CAY10573 demonstrates stronger binding and functional activity for PPARγ than the antidiabetic compound rosiglitazone (IC50 = 92 nM; EC50 = 220 nM).

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