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安捷凯生物医药，安捷凯化学
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  2. Casein Kinase
  3. CAY10578
  • CAY10578
CAY10578的可视化放大

CAY10578

A potent and selective CK2 inhibitor

原价
￥262-4675
价格
￥ 210-3740
CAY10578的二维码

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  • 库存: 现货
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  • 货号: ajci70596
  • CAS: 19231-60-8
  • 别名:
  • 分子式: C10H3I4NO4
  • 分子量: 708.8
  • 纯度: >98%
  • 溶解度: DMF: 10 mg/ml,DMF:PBS (pH 7.2) 1:5: 0.15 mg/ml,DMSO: 5 mg/ml
  • 储存: Store at -20°C
  • 库存: 现货

Background

Casein Kinase 2 (CK2) is a constitutive protein kinase involved in many signal transduction pathways. CK2 is known to negatively regulate apoptosis, and its activity is increased in many proliferating tissues and tumors, which lends promise as an anticancer drug target. CAY10578 is a potent inhibitor of CK2 with an IC50 value of 0.3 µM. This compound is ATP competitive, displaying a Ki value of 0.2 µM and only minimally inhibits the activities of other protein kinases (e.g., GSK3, Cdk5, and MSK1).

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