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  • XMD-17-51 Trifluoroacetate
XMD-17-51 Trifluoroacetate的可视化放大

XMD-17-51 Trifluoroacetate

XMD-17-51 Trifluoroacetate 是一种能够调节蛋白激酶的嘧啶并二氮杂酮化合物。

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XMD-17-51 Trifluoroacetate的二维码
  • 库存: 现货
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  • 包装
    价格
    促销价
    数量
  • 5mg
    ¥2062.00
    1650.00
    - +
  • 10mg
    ¥3225.00
    2580.00
    - +
  • 25mg
    ¥6462.00
    5170.00
    - +
已选 0 0
金额: ¥0.00
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  • 货号: ajcx11632
  • CAS: N/A
  • 别名:
  • 分子式: C23H25F3N8O3
  • 分子量: 518.49
  • 纯度: >98%
  • 溶解度: DMSO : ≥ 150 mg/mL (289.30 mM)
  • 储存: Store at -20°C
  • 库存: 现货

Background

XMD-17-51 Trifluoroacetate is a pyrimido-diazepinone compound that is able to modulate protein kinases.


XMD-17-51 Trifluoroacetate is a pyrimido-diazepinone compound that is able to modulate protein kinases, including MPS1 (TTK), ERK5 (BMK1, MAPK7), polo kinase 1, 2, 3, or 4, Ack1, Ack2, Abl, DCAMKL1, ABL1, Abl mutants, DCAMKL2, ARK5, BRK, MKNK2, FGFR4, TNK1, PLK, ULK2, PLK, PRKD1, PRKD2, PRKD3, ROS1, RPS6KA6, TAOK1, TAOK3, TNK2, Bcr-Abl, GAK, cSrc, TPR-Met, Tie2, MET, FGFR3, Aurora, Axl, Bmx, BTK, c-kit, CHK2, Flt3, MST2, p70S6K, PDGFR, PKB, PKC, Raf, ROCK-H, Rsk1, SGK, TrkA, TrkB and TrkC, and can be used in the treatment of various diseases, disorders or conditions[1].

参考文献:
[1]. WO 2014145909 A2.

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