UAAcrosslinker1可充当pylRS/tRNA对的底物,能够掺入靶蛋白中。
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UAA crosslinker 1 act as substrates for pylRS/tRNA pair that enable its incorporation into a target protein.
[1]. VanBrunt MP, et al. Genetically Encoded Azide Containing Amino Acid in Mammalian Cells Enables Site-Specific Antibody-Drug Conjugates Using Click Cycloaddition Chemistry. Bioconjug Chem. 2015 Nov 18;26(11):2249-60.