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AGI-25696是蛋氨酸腺苷转移酶(MATA2)抑制剂,对研究癌症有用。AGI-25696阻断体内MTAP缺失的肿瘤的生长。
AGI-25696 is a methionine adenosyltransferase 2A (MATA2 ) inhibitors useful for treatment of cancer. AGI-25696 blocks growth of MTAP-deleted tumors in vivo.
[1]. Agios. Targeting MAT2A in MTAP-deleted Cancers. Presented at the American Association for Cancer Research (AACR) Annual Meeting, April 14-18, 2018, Chicago, IL, USA
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