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ElacestrantSenantiomer是elacestrant的低活性对映体。Elacestrant(RAD1901)是有选择性和口服活性的雌激素受体(ER)的降解剂,对ERα和ERβ的IC50值分别为48和870nM。
Elacestrant S enantiomer is an low activity enantiomer of elacestrant. Elacestrant (RAD1901) is a selective and orally available estrogen receptor (ERR) degrader with IC50 values of 48 and 870 nM for ERα and ERβ, respectively.
[1]. Garner F, et al. RAD1901: a novel, orally bioavailable selective estrogen receptor degrader that demonstrates antitumor activity in breast cancer xenograft models. Anticancer Drugs. 2015 Oct;26(9):948-56.
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