Elacestrant S enantiomer (RAD1901 S enantiomer)
ElacestrantSenantiomer是elacestrant的低活性对映体。Elacestrant(RAD1901)是有选择性和口服活性的雌激素受体(ER)的降解剂，对ERα和ERβ的IC50值分别为48和870nM。
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包装价格促销价数量
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1mg￥1612.001290.00- +
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5mg￥3737.002990.00- +
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10mg￥5350.004280.00- +
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50mg￥15887.0012710.00- +
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- 货号: ajcx13322
- CAS: N/A
- 别名:
- 分子式: C30H38N2O2
- 分子量: 458.63
- 纯度: ＞98%
- 溶解度: Soluble in DMSO
- 储存: Store at -20°C
- 库存: 现货
Background
Elacestrant S enantiomer is an low activity enantiomer of elacestrant. Elacestrant (RAD1901) is a selective and orally available estrogen receptor (ERR) degrader with IC50 values of 48 and 870 nM for ERα and ERβ, respectively.
[1]. Garner F, et al. RAD1901: a novel, orally bioavailable selective estrogen receptor degrader that demonstrates antitumor activity in breast cancer xenograft models. Anticancer Drugs. 2015 Oct;26(9):948-56.
