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Seco-Duocarmycin SA 是一种高效的 DNA 烷化剂 (DNA alkylator),可作用做抗体-药物偶联物 (ADC) 的毒素部分。
Seco-Duocarmycin SA is a highly potent DNA alkylator, and is used as an ADC cytotoxin[1].
[1]. Lutz F. Tietze, et al. A Concise and Efficient Synthesis of seco-Duocarmycin SA. European Journal of Organic Chemistry 2003 (3), 562-566.
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