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Vat-Cit-PAB-Monomethyl Dolastatin 10 是抗体-药物偶联物的一部分,由 Monomethyl Dolastatin 10 (一种有效的微管蛋白抑制剂) 和 ADC linker Vat-Cit-PAB 连接而成。
Vat-Cit-PAB-Monomethyl Dolastatin 10 is a drug-linker conjugate for ADC with potent antitumor activity by using Monomethyl Dolastatin 10 (a potent tubulin inhibitor), linked via the ADC linker Vat-Cit-PAB.
[1]. Chudasama V, et al. Recent advances in the construction of antibody-drug conjugates. Nat Chem. 2016 Feb;8(2):114-9.
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