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ONC206

ONC206 is a selective antagonist of dopamine D2-like receptors (DRD2/3/4) with broad-spectrum anti-tumor activity.

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ONC206的二维码
  • 库存: 现货
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  • 1mg
    ¥437.00
    350.00
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  • 5mg
    ¥1112.00
    890.00
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  • 10mg
    ¥1950.00
    1560.00
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  • 25mg
    ¥3300.00
    2640.00
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  • 50mg
    ¥6037.00
    4830.00
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  • 100mg
    ¥10662.00
    8530.00
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  • 货号: ajcx15654
  • CAS: 1638178-87-6
  • 别名:
  • 分子式: C23H22F2N4O
  • 分子量: 408.44
  • 纯度: >98%
  • 溶解度: DMSO: 100 mg/mL (244.83 mM)
  • 储存: Store at -20°C
  • 库存: 现货

Background

ONC206 is a selective antagonist of dopamine D2-like receptors (DRD2/3/4) with broad-spectrum anti-tumor activity.


ONC206 is a ClpP agonist regarding the requirement of high doses (50–130?mg/kg) to achieve in vivo efficacy. [2]


[1] Varun Vijay Prabhu, et al. Cancer Res 2017;77(13 Suppl):Abstract nr 4147A. [2] Fennell EMJ, et al. Pharmacol Res Perspect. 2022 Aug;10(4):e00993.

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