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  • CTAP (trifluoroacetate salt)
CTAP (trifluoroacetate salt)的可视化放大

CTAP (trifluoroacetate salt)

An antagonist of the μ opioid receptor

原价
￥2400-2400
价格
￥ 1920-1920
CTAP (trifluoroacetate salt)的二维码

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  • 库存: 现货
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  • 货号: ajcx18292
  • CAS: N/A
  • 别名:
  • 分子式: C51H69N13O11S2?XCF3COOH
  • 分子量: 1104.3
  • 纯度: >98%
  • 溶解度: Water: soluble
  • 储存: Store at -20°C
  • 库存: 现货

Background

CTAP is a water soluble, cyclic octapeptide which acts as a receptor antagonist that is selective for the µ opioid receptor (IC50 = 3.5 nM) over the δ receptor (IC50 = 4,500 nM). It is a poor antagonist of the somatostatin receptor (IC50 = 14.3 μM). CTAP is at least 10-fold more potent than naltrexone as an antagonist of diverse compounds which have antinociceptive effects through the µ opioid receptor. It resists enzymatic metabolism in the blood and enters the brain and cerebrospinal fluid.

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