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- Ribosomal S6 Kinase (RSK)
- Bilaid A1
Bilaid A1
A tetrapeptide
此产品仅用于科学研究，我们不为任何个人用途提供产品和服务
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包装价格促销价数量
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1mg￥4000.003200.00- +
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5mg￥14862.0011890.00- +
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- 货号: ajcx21806
- CAS: 2393866-02-7
- 别名: H-FVVF-NH2, H-L-Phe-D-Val-L-Val-D-Phe-NH2
- 分子式: C28H39N5O4
- 分子量: 509.6
- 纯度: ＞98%
- 溶解度:
- 储存: Store at -20°C
- 库存: 现货
Background
Bilaid A1 is a tetrapeptide agonist of the µ-opioid receptor (Ki = 750 nM in HEK293 cell membranes expressing the human receptor) and a derivative of bilaid A .1 It inhibits forskolin-induced cAMP accumulation by 47% in HEK293 cells expressing the human µ-opioid receptor when used at a concentration of 10 µM.
1.Dekan, Z., Sianati, S., Yousuf, A., et al.A tetrapeptide class of biased analgesics from an Australian fungus targets the µ-opioid receptorProc. Natl. Acad. Sci. USA116(44)22353-22358(2019)
