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- 5-HT Receptor
- RS 127445 hydrochloride
RS 127445 hydrochloride
A 5-HT2B receptor antagonist
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包装价格促销价数量
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10mg￥1000.00800.00- +
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50mg￥4337.003470.00- +
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- 货号: ajcx26798
- CAS: 199864-86-3
- 别名: 4-(4-氟-1-萘基)-6-(1-甲基乙基)-2-嘧啶胺盐酸盐
- 分子式: C17H16FN3.HCl
- 分子量: 317.79
- 纯度: ＞98%
- 溶解度: Soluble in DMSO
- 储存: Store at -20°C
- 库存: 现货
Background
High affinity 5-HT2B receptor antagonist (pKi = 9.5). Displays 1000-fold selectivity for 5-HT2B with good bioavailability.
Bonhaus et al (1999) RS-127445: a selective, high affinity, orally bioavailable 5-HT2B receptor antagonist. Br.J.Pharmacol. 127 1075 PMID:10455251 |Callebert et al (2006) Evidence for a control of plasma serotonin levels by 5-Hydroxytryptamine2B receptors in mice. J.Pharmacol.Exp.Ther. 317 724 PMID:16461587
