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5-HT1Amodulator2hydrochloride是8-OH-DPAT的一种衍生物,5-HT1Amodulator2hydrochloride是5-HT1A的调节剂,与5-HT1A结合的Ki值为53nM。
5-HT1A modulator 2 hydrochloride, a derivative of 8-OH-DPAT , is a modulator of 5-HT1A with a Ki of 53 nM for 5-HT1A binding[1].
[1]. Naiman, N.,et al. 2-(Alkylamino)tetralin derivatives: interaction with 5-HT1A serotonin binding sites. Journal of Medicinal Chemistry, 1989;32(1), 253-256.
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