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  • Lobaplatin
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Lobaplatin

Lobaplatin (D-19466) is a third-generation platinum anti-neoplastic agent. It is a platinum complex with DNA alkylating activity.DMSO is not recommended to dissolve platinum-based drugs, which can easily lead to drug inactivation.

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¥1212-17100
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970-13680
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  • 货号: ajcx30938
  • CAS: 135558-11-1
  • 别名: 络铂; D-19466
  • 分子式: C9H18N2O3Pt
  • 分子量: 397.33
  • 纯度: >98%
  • 溶解度: Water: ≥ 50 mg/mL (125.84 mM; DMSO can inactivate Lobaplatin's activity)
  • 储存: Store at -20°C
  • 库存: 现货

Background

Lobaplatin (D-19466) is a third-generation platinum anti-neoplastic agent. It is a platinum complex with DNA alkylating activity.DMSO is not recommended to dissolve platinum-based drugs, which can easily lead to drug inactivation.


Lobaplatin has excellent anticancer activity in vivo against a number of murine experimental tumors, including a cisplatin-resistant P388 line. [1]


[1] Voegeli R,et al.J Cancer Res Clin Oncol.1990;116(5):439-42. [2] Matthew D Hall, et al. Cancer Res. 2014 Jul 15;74(14):3913-22.

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