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Lobaplatin (D-19466) is a third-generation platinum anti-neoplastic agent. It is a platinum complex with DNA alkylating activity.DMSO is not recommended to dissolve platinum-based drugs, which can easily lead to drug inactivation.
Lobaplatin (D-19466) is a third-generation platinum anti-neoplastic agent. It is a platinum complex with DNA alkylating activity.DMSO is not recommended to dissolve platinum-based drugs, which can easily lead to drug inactivation.
Lobaplatin has excellent anticancer activity in vivo against a number of murine experimental tumors, including a cisplatin-resistant P388 line. [1]
[1] Voegeli R,et al.J Cancer Res Clin Oncol.1990;116(5):439-42. [2] Matthew D Hall, et al. Cancer Res. 2014 Jul 15;74(14):3913-22.
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