S961 acetate

S961acetate是一种高亲和力的胰岛素受体(insulinreceptor,IR)拮抗剂，对HIR-A，HIR-B和人胰岛素样生长因子I受体(HIGF-IR)的IC50分别为0.048，0.027和630nM。

原价

￥3262-3262

价格

￥ 2610-2610

所有产品仅用于科学研究，我们不为任何个人用途提供产品和服务

询价有惊喜，量大更优惠

库存: 现货

可选包装 >>>

首页

产品引用

货号: ajcx31988
CAS: N/A
别名:
分子式: C213H301N55O72S2
分子量: 4864.18
纯度: >98%
溶解度: DMSO : 12.5 mg/mL?(2.57 mM;?) Water : 1.79 mg/mL?(0.37 mM;?ultrasonic and adjust pH to 8 with NaOH)
储存: Store at -20°C
库存: 现货

Background

S961 acetate is an high-affinity and selective insulin receptor (IR) antagonist with IC50s of 0.048, 0.027, and 630 nM for HIR-A, HIR-B, and human insulin-like growth factor I receptor (HIGF-IR) in SPA-assay, respectively[1].

S961 also shows high-affinity to Rat IR and Pig IR with IC50s of 0.056 nM and 0.084 nM in PEG-assay, respectively[1].

[1]. Sch?ffer L, et al. A novel high-affinity peptide antagonist to the insulin receptor. Biochem Biophys Res Commun. 2008 Nov 14;376(2):380-3.

动态评分

0.0

没有评分数据

没有评价数据