- 首页
- HDAC (Histone deacetylases)
- LSD1/HDAC6-IN-1
LSD1/HDAC6-IN-1
LSD1/HDAC6-IN-1 是一种具有口服活性的组蛋白去甲基化酶 LSD1 和组蛋白去乙酰酶 HDAC6 (LSD1/HDAC6) 双重抑制剂，具有抗肿瘤活性。LSD1/HDAC6-IN-1 可用于多发性骨髓瘤 (MM) 的研究。
此产品仅用于科学研究，我们不为任何个人用途提供产品和服务
-
包装价格促销价数量
-
5mg￥4200.003360.00- +
-
10mg￥6737.005390.00- +
-
25mg￥13350.0010680.00- +
已选
0
种
0
瓶
金额:
￥0.00
首页
收藏
- 货号: ajcx33714
- CAS: 2738306-38-0
- 别名:
- 分子式: C25H33N3O2
- 分子量: 407.55
- 纯度: ＞98%
- 溶解度:
- 储存: Store at -20°C
- 库存: 现货
Background
LSD1/HDAC6-IN-1 is an orally active dual inhibitor of lysine specific demethylase 1(LSD1)/Histone deacetylase 6 (HDAC6), with anti-tumor activity. LSD1/HDAC6-IN-1 can be used for the research of multiple myeloma (MM)[1].
LSD1/HDAC6-IN-1 shows superior potency in multiple MM lines[1].
LSD1/HDAC6-IN-1 is efficacy in the MM.1S xenograft model[1].
[1]. M Naveen Sadhu, et al. Novel dual LSD1/HDAC6 inhibitors for the treatment of multiple myeloma. Bioorg Med Chem Lett. 2020 Dec 24;34:127763.
