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  • Stafia-1-dipivaloyloxymethyl ester
Stafia-1-dipivaloyloxymethyl ester的可视化放大

Stafia-1-dipivaloyloxymethyl ester

Stafia-1-dipivaloyloxymethyl ester (compound 27) 是有效的、选择性的STAT5a 抑制剂。

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¥4850-17625
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3880-14100
Stafia-1-dipivaloyloxymethyl ester的二维码

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  • 货号: ajcx35220
  • CAS: 2582755-72-2
  • 别名:
  • 分子式: C37H48FO13P
  • 分子量: 750.74
  • 纯度: >98%
  • 溶解度: DMSO : 100 mg/mL (133.20 mM; Need ultrasonic)
  • 储存: Store at -20°C
  • 库存: 现货

Background

Stafia-1-dipivaloyloxymethyl ester (compound 27, 0-200 μM) decreases pSTAT5a expression significantly, and has no obvious inhibition on pSTAT5b[1].


Stafia-1-dipivaloyloxymethyl ester (compound 27, 0-200 μM) decreases pSTAT5a expression significantly, and has no obvious inhibition on pSTAT5b[1].


[1]. Kalaiselvi Natarajan, et al. Stafia-1: A STAT5a-Selective Inhibitor Developed via Docking-Based Screening of in Silico O-Phosphorylated Fragments. Chemistry. 2020 Jan 2;26(1):148-154.

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