Trifluoperazine D8 是 Trifluoperazine 的氘代物。Trifluoperazine 是一种抗精神病药物吩噻嗪类药物,是一种选择性的 α1-肾上腺素能受体拮抗剂。Trifluoperazine 也是一种有效的多巴胺 D2 受体抑制剂。
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Trifluoperazine D8 is a deuterium labeled Trifluoperazine. Trifluoperazine is an antipsychotic phenothiazine agent and a selective α1-adrenergic receptor antagonist. Trifluoperazine is also a potent dopamine D2 receptor inhibitor [1][2].
[1]. Huerta-Bahena J, et al. Trifluoperazine and chlorpromazine antagonize alpha 1- but not alpha2- adrenergic effects. Mol Pharmacol. 1983 Jan;23(1):67-70.
[2]. Marques LO, et al. Trifluoperazine for schizophrenia. Cochrane Database Syst Rev. 2004;(1):CD003545.
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