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CC-99677

CC-99677 是一种有效的、共价的、不可逆的丝裂原活化蛋白 (MAP) 激酶活化蛋白激酶 -2 (MK2)通路抑制剂,在生化(IC50=156.3 nM) 和细胞基础检测 (EC50=89 nM) 中均有作用。CC-99677 来自专利 WO2020236636,化合物 1。

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CC-99677的二维码
  • 库存: 现货
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  • 包装
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    促销价
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  • 5mg
    ¥9175.00
    7340.00
    - +
  • 10mg
    ¥13887.00
    11110.00
    - +
已选 0 0
金额: ¥0.00
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  • 货号: ajcx35686
  • CAS: 1887069-10-4
  • 别名:
  • 分子式: C22H20ClN5O3S
  • 分子量: 469.94
  • 纯度: >98%
  • 溶解度:
  • 储存: Store at -20°C
  • 库存: 现货

Background

CC-99677 is a potent, covalent, and irreversible inhibitor of the mitogen-activated protein (MAP) kinase-activated protein kinase-2 (MK2) pathway in both biochemical (IC50=156.3 nM) and cell based assays (EC50=89 nM). CC-99677 is extracted from patent WO2020236636, compound 1[1].


CC-99677 is a potent, covalent, and irreversible inhibitor of the mitogen-activated protein (MAP) kinase-activated protein kinase-2 (MK2) pathway in both biochemical (IC50=156.3 nM) and cell based assays (EC50=89 nM)[1].


[1]. WO2020236636

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