G-Protein antagonist peptide TFA

G-Protein antagonist peptide TFA 是一种截短的 substance P 相关肽，与受体竞争 G 蛋白结合。G-Protein antagonist peptide TFA 抑制重组磷脂囊泡中 M2 毒蕈碱胆碱能受体 (M2 mAChR) 激活 Gi 或 Go 或 β 肾上腺素能受体激活 Gs。

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库存: 现货

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1mg

￥1625.00

1300.00

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5mg

￥4312.00

3450.00

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10mg

￥6900.00

5520.00

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已选 0 种 0 瓶

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货号: ajcx36322
CAS: N/A
别名:
分子式: C59H65F3N12O11S
分子量: 1207.28
纯度: >98%
溶解度: DMSO : 50 mg/mL (41.42 mM; Need ultrasonic)
储存: -20°C, away from moisture
库存: 现货

Background

G-Protein antagonist peptide TFA is a truncated substance P-related peptide, competes with receptor for G protein binding. G-Protein antagonist peptide TFA inhibits the activation of Gi or Go by M2 muscarinic cholinergic receptor (M2 mAChR) or of Gs by beta-adrenergic receptor in the reconstituted phospholipid vesicles, assayed by receptor-promoted GTP hydrolysis[1].

[1]. Mukai H, et al. G protein antagonists. A novel hydrophobic peptide competes with receptor for G protein binding. J Biol Chem. 1992;267(23):16237-16243.