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  • Mc-Alanyl-Alanyl-Asparagine-PAB-MMAE
Mc-Alanyl-Alanyl-Asparagine-PAB-MMAE的可视化放大

Mc-Alanyl-Alanyl-Asparagine-PAB-MMAE

Mc-Alanyl-Alanyl-Asparagine-PAB-MMAE (compound S6) 是一种有效的抗癌剂 (anticancer agent),它可被肿瘤微环境特异性激活。Mc-Alanyl-Alanyl-Asparagine-PAB-MMAE 可抑制小鼠肿瘤生长 (信息来自专利 CN104147612A)。

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Mc-Alanyl-Alanyl-Asparagine-PAB-MMAE的二维码
  • 库存: 现货
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  • 包装
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  • 5mg
    ¥8412.00
    6730.00
    - +
  • 10mg
    ¥13350.00
    10680.00
    - +
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  • 货号: ajcx39804
  • CAS: 1638970-46-3
  • 别名:
  • 分子式: C67H101N11O16
  • 分子量: 1316.58
  • 纯度: >98%
  • 溶解度: DMSO : 180 mg/mL (136.72 mM; Need ultrasonic)
  • 储存: 4°C, protect from light, stored under nitrogen
  • 库存: 现货

Background

Mc-Alanyl-Alanyl-Asparagine-PAB-MMAE (compound S6) is a potent anticancer agent, which can be specific activated by tumor microenvironment. Mc-Alanyl-Alanyl-Asparagine-PAB-MMAE can suppress tumor growth in mice (extracted from patent CN104147612A)[1].


Mc-Alanyl-Alanyl-Asparagine-PAB-MMAE (compound S6) (26.2 micro-rubbing/kg, IV, weekly for 4 weeks) suppresses tumor growth in mice bearing Panc-1 tumor[1].


[1]. Liu Chen, et al. Tumor microenvironment specific activated micromolecular targeted conjugate and application thereof. CN104147612A.

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