Ritanserin

A potent 5-HT2A receptor antagonist

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库存: 现货

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数量
5mg

￥600.00

480.00

- +
10mg

￥1025.00

820.00

- +
25mg

￥2200.00

1760.00

- +

已选 0 种 0 瓶

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货号: ajci12008
CAS: 87051-43-2
别名: 利坦丝林,R 55667
分子式: C27H25F2N3OS
分子量: 477.57
纯度: >98%
溶解度: DMF: 30 mg/ml,DMSO: 12.5 mg/ml,Ethanol: 2.5 mg/ml
储存: Store at -20°C
库存: 现货

Background

Ritanserin (R 55667) is a highly potent, relatively selective, orally active, long acting antagonist of 5-HT2 receptor, with an IC50 of 0.9 nM, less active on Histamine H1, Dopamine D2, Adrenergic α1, Adrenergic α2 receptors[1].

Ritanserin (R 55667) is a highly potent, relatively selective, long acting antagonist of 5-HT2 receptor, with an IC50 of 0.9 nM, less active on Histamine-H1 (IC50, 35 nM), Dopamine-D2 (IC50, 70 nM), Adrenergic-α1 (IC50, 97 nM), Adrenergic-α2 receptor (IC50, 150 nM)[1].

参考文献:
[1]. Leysen JE, et al. Receptor-binding properties in vitro and in vivo of ritanserin: A very potent and long acting serotonin-S2 antagonist. Mol Pharmacol. 1985 Jun;27(6):600-11.