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  • Todralazine (hydrochloride)
Todralazine (hydrochloride)的可视化放大

Todralazine (hydrochloride)

A β2-adrenergic receptor antagonist

原价
¥1437-5050
价格
1150-4040
Todralazine (hydrochloride)的二维码

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  • 库存: 现货
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  • 货号: ajci20896
  • CAS: 3778-76-5
  • 别名: 盐酸托屈嗪,Ecarazine hydrochloride
  • 分子式: C11H12N4O2.HCl
  • 分子量: 268.7
  • 纯度: >98%
  • 溶解度: DMF: 5 mg/ml,DMSO: 10 mg/ml,DMSO:PBS (pH 7.2) (1:1): 0.5 mg/ml,Ethanol: 1 mg/ml,PBS (pH 7.2): slightly
  • 储存: Store at -20°C
  • 库存: 现货

Background

Todralazine (hydrochloride) is a β2-adrenergic receptor antagonist with peripheral vasodilator activity. Administration of todralazine (5 uM) to pre-larval zebrafish led to hematopoietic cell expansion and protection from ionizing radiation. It inhibited histone acetylation in vitro and, long-term (4 months), but not short-term (1 month), treatment in mice (3 mg/day) impaired hepatocyte histone acetylation and liver regeneration.

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