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  2. RIP kinase
  3. (±)-WIN 55,212 (mesylate)
  • (±)-WIN 55,212 (mesylate)
(±)-WIN 55,212 (mesylate)的可视化放大

(±)-WIN 55,212 (mesylate)

A racemic mixture of (+)-WIN 55,212-2 and (?)-WIN 55,212-3

原价
￥612-4925
价格
￥ 490-3940
(±)-WIN 55,212 (mesylate)的二维码

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  • 库存: 现货
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  • 货号: ajci67612
  • CAS: 137795-17-6
  • 别名:
  • 分子式: C27H26N2O3?CH3SO3H
  • 分子量: 522.6
  • 纯度: >98%
  • 溶解度: DMF: 30 mg/ml,DMSO: 30 mg/ml,DMSO:PBS(pH 7.2) (1:2): 0.25 mg/ml,Ethanol: 5 mg/ml
  • 储存: Store at -20°C
  • 库存: 现货

Background

(±)-WIN 55,212-2 is a potent aminoalkylindole cannabinoid (CB) receptor agonist with a Ki value of 62.3 and 3.3 nM for human recombinant central cannabinoid (CB1) and peripheral cannabinoid (CB2) receptors, respectively. In contrast, the enantiomer (-)-WIN 55,212-3 acts a partial inverse agonist at CB1 (pIC50 = 5.5) and as a competitive neutral antagonist of CB2, reversing the inverse agonism evoked by SR 144528 (pEC50 = 5.3). (+)-WIN 55,212 (mesylate) is a mixture of the two enantiomers, (+)-WIN 55,212-2 and (-)-WIN 55,212-3.

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