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CDK1-IN-2 是一种 CDK1 抑制剂 (IC50: 5.8 μM)。
CDK1-IN-2 is a CDK1 inhibitor (IC50: 5.8 μM)[1].
CDK1-IN-2 ("CDK1 inhibitor 1", 0-19.8 μM, 24 h) arrests HCT-116 cells in G2/M phase[1].
[1]. Jorda R, et al. How Selective Are Pharmacological Inhibitors of Cell-Cycle-Regulating Cyclin-Dependent Kinases? J Med Chem. 2018 Oct 25;61(20):9105-9120.
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