安捷凯生物医药
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  • Eletriptan
Eletriptan的可视化放大

Eletriptan

An agonist of 5-HT1B and 5-HT1D receptors

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Eletriptan的二维码
  • 库存: 现货
可选规格
  • 包装
    价格
    促销价
    数量
  • 1mg
    ￥1337.00
    1070.00
    - +
  • 5mg
    ￥2687.00
    2150.00
    - +
  • 10mg
    ￥4675.00
    3740.00
    - +
  • 50mg
    ￥19825.00
    15860.00
    - +
已选 0 种 0 瓶
金额: ￥0.00
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使用我司产品发表的文章

  • 货号: ajci71430
  • CAS: 143322-58-1
  • 别名: 依来曲普坦,UK-116044
  • 分子式: C22H26N2O2S
  • 分子量: 382.5
  • 纯度: >98%
  • 溶解度: DMF: 10 mg/ml,DMF:PBS(pH 7.2)(1:1): 0.5 mg/ml,DMSO: 10 mg/ml,Ethanol: 0.1 mg/ml
  • 储存: Store at -20°C
  • 库存: 现货

Background

Eletriptan is an agonist of the serotonin (5-HT) receptor types 5-HT1B and 5-HT1D. It inhibits forskolin-induced cAMP accumulation in and induces vasoconstriction of isolated rabbit common carotid artery rings (pD2s = 7.6 and 4.9, respectively), an effect that can be blocked by the 5-HT1B antagonist SB216641 but not the 5-HT1D antagonist BRL15572. Eletriptan preferentially induces constriction of isolated human cerebral over coronary arteries (EC50s = 15.8 and 1,995 nM, respectively). Formulations containing eletriptan have been used in the treatment of migraine headache.

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