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  • β-Amino Acid Imagabalin Hydrochloride (PD-0332334)
β-Amino Acid Imagabalin Hydrochloride (PD-0332334)的可视化放大

β-Amino Acid Imagabalin Hydrochloride (PD-0332334)

β-Amino Acid Imagabalin Hydrochloride (PD-0332334) (PD-0332334) 是 α2&#948 的配体;电压依赖性钙通道的亚基。

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β-Amino Acid Imagabalin Hydrochloride (PD-0332334)的二维码
  • 库存: 现货
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  • 1mg
    ¥15250.00
    12200.00
    - +
  • 5mg
    ¥34325.00
    27460.00
    - +
  • 10mg
    ¥58387.00
    46710.00
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  • 20mg
    ¥103012.00
    82410.00
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  • 货号: ajce46738
  • CAS: 610300-00-0
  • 别名: PD-0332334
  • 分子式: C9H20ClNO2
  • 分子量: 209.71
  • 纯度: >98%
  • 溶解度: Soluble in DMSO
  • 储存: Store at -20°C
  • 库存: 现货

Background

β-Amino Acid Imagabalin Hydrochloride (PD-0332334) is a ligand for the α2δ subunit of the voltage-dependent calcium channel.


β-Amino Acid Imagabalin Hydrochloride had been in phase III clinical trials for the treatment of generalised anxiety disorders. However, this research has been discontinued[2]. β-Amino Acid Imagabalin Hydrochloride had been also in phase I clinical trials for the treatment of chronic kidney disease[3].


[1]. Birch M, et al. A Simplified Process for the Manufacture of Imagabalin Hydrochloride (PD-0332334), an α2δ-Ligand for the Treatment of Generalised Anxiety Disorder. Org. Process Res. Dev., 2011, 15 (6), pp 1358-1364

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