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ROCK-IN-1是一种有效的ROCK抑制剂,能够抑制ROCK2的活性,IC50值为1.2nM。
ROCK-IN-1 is a potent inhibitor of ROCK, with an IC50 of 1.2 nM for ROCK2.
ROCK-IN-1 shows potent cellular efficacy, with an EC50 of 200 nM[1].
[1]. Boland S, et al. 3-[2-(Aminomethyl)-5-[(pyridin-4-yl)carbamoyl]phenyl] benzoates as soft ROCK inhibitors. Bioorg Med Chem Lett. 2013 Dec 1;23(23):6442-6.
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