ZK-90055 hydrochloride

ZK-90055hydrochloride是β2肾上腺素能受体(β2adrenergicreceptor)激动剂。

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库存: 现货

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促销价

数量
1mg

￥5987.00

4790.00

- +
5mg

￥11987.00

9590.00

- +
10mg

￥21287.00

17030.00

- +
20mg

￥36862.00

29490.00

- +

已选 0 种 0 瓶

金额: ￥0.00

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Background

ZK-90055 hydrochloride is a β2 adrenergic receptor agonist.

Contrasting a pro-drug, a soft-drug is active per se when given locally but is rapidly inactivated when it reaches the general circulation. Thus, a long duration of action at a minimum of systemic side effects may be achieved after inhalation of a h2-agonist designed in this way. One such example is ZK-90055, an indol derivative with a hydrolysable ester bond on the ring system. The development of ZK-90055 is stopped before clinical trials are commenced[2].

[1]. Waldeck B, et al. beta-Adrenoceptor agonists after terbutaline. Pharmacol Toxicol. 1995;77 Suppl 3:25-9. [2]. Waldeck B, et al. Beta-adrenoceptor agonists and asthma--100 years of development. Eur J Pharmacol. 2002 Jun 7;445(1-2):1-12.