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JAK3-IN-7是一种有效的选择性JAK3抑制剂,详细信息请参考专利文献WO2011013785A1中表1-1中的化合物1和2,IC50<0.01μM。
JAK3-IN-7 is a potent and selective JAK3 inhibitor extracted from patent WO2011013785A1, has an IC50 of <0.01 μM.
[1]. NOJI, Satoru, et al. NITROGEN-CONTAINING SPIRO-RING COMPOUND AND MEDICINAL USE OF SAME. WO2011013785A1.
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