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  • Niraparib metabolite M1 (Niraparib carboxylic acid metabolite M1)
Niraparib metabolite M1 (Niraparib carboxylic acid metabolite M1)的可视化放大

Niraparib metabolite M1 (Niraparib carboxylic acid metabolite M1)

Niraparib 代谢物 M1 (Niraparib carboxy acid metabolite M1) 是 niraparib 的代谢物,后者作为一种新型聚 (ADP-核糖) 聚合酶 (PARP) 抑制剂。

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Niraparib metabolite M1 (Niraparib carboxylic acid metabolite M1)的二维码

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  • 货号: ajce51146
  • CAS: 1476777-06-6
  • 别名: 尼拉帕尼代谢物; Niraparib carboxylic acid metabolite M1; M1 metabolite of niraparib
  • 分子式: C19H19N3O2
  • 分子量: 321.37
  • 纯度: >98%
  • 溶解度: DMSO : ≥ 100 mg/mL (311.17 mM)
  • 储存: Store at -20°C
  • 库存: 现货

Background

Niraparib metabolite M1 is a metabolite of niraparib, and the latter one acts as a novel poly(ADP-Ribose) polymerase (PARP) inhibitor.


Niraparib metabolite M1 has the validation in plasma and urine for the support of clinical studies such as the mass balance study and the absolute bioavailability study[1].


[1]. van Andel L, et al. Liquid chromatography-tandem mass spectrometry assay for the quantification of niraparib and its metabolite M1 in human plasma and urine. J Chromatogr B Analyt Technol Biomed Life Sci. 2016 Nov 19;1040:14-21.

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