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CB2R-IN-1是一种有效的cannabinoidCB2受体反向激动剂,Ki为0.9nM。
CB2R-IN-1 is a potent cannabinoid CB2 receptor inverse agonist with a Ki of 0.9 nM.
CB2R-IN-1 (Compound 37) is a potent cannabinoid CB2 receptor ligand (Ki=0.9 nM) with excellent selectivity over the CB1 receptor (Ki=8259.3 nM)[1].
[1]. Tong L, et al. Expansion of SAR studies on triaryl bis sulfone cannabinoid CB2 receptor ligands. Bioorg Med Chem Lett. 2010 Nov 15;20(22):6785-9.
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