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DSP-2230 是选择性的 Nav1.7/Nav1.8 通道阻断剂。
DSP-2230 is a selective Nav1.7/Nav1.8 blocker[1][2]. Nav1.7/Nav1.8[1]
[1]. Bagal SK, et al. Voltage gated sodium channels as drug discovery targets. Channels (Austin). 2015;9(6):360-6. [2]. Sara Sabina Hadida-Ruah, et al. Sulfonamides as modulators of sodium channels.
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