安捷凯在线客服
- 客服:
- 电话: 13061953619
- 微信:
IDH1 Inhibitor 2 是有效的IDH1 抑制剂,通过对 His315的共价修饰发挥作用,其IC50 值为110 nM。
IDH1 Inhibitor 2 is a potent IDH1 inhibitor via a direct covalent modification of His315, with an IC50 of 110 nM[1]. IC50: 110 nM (IDH1)[1].
[1]. Jakob CG, et al. Novel Modes of Inhibition of Wild-Type Isocitrate Dehydrogenase 1 (IDH1): Direct Covalent Modification of His315. J Med Chem. 2018 Aug 9;61(15):6647-6657.
动态评分
0.0