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A JAK1 inhibitor
Itacitinib is an inhibitor of JAK1.1 It is greater than 20- and 200-fold selective for JAK1 over JAK2 and JAK3, respectively.
1.Norman, P.Selective JAK inhibitors in development for rheumatoid arthritisExpert Opin. Investig. Drugs23(8)1067-1077(2014)
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