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Taranabant (1R,2R)stereoisomer 是 Taranabant 的 R 型对映异构体。Taranabant 是有效的选择性 cannabinoid 1 (CB1) 受体反向激动剂。
Taranabant (1R,2R)stereoisomer is the R-enantiomer of Taranabant. Taranabant is a highly potent and selective cannabinoid 1 (CB1) receptor inverse agonist.
[1]. William K. Hagmann, et al. Substituted amides active at the cannabinoid-1 receptor. WO 2004048317 A1.
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