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Trans (2,3)-Dihydrotetrabenazine, 是抗精神病药物Tetrabenazine的体内代谢物,能够抑制囊泡单胺转运体 2 (VMAT2)。
Trans (2,3)-Dihydrotetrabenazine, a metabolite of Tetrabenazine, shows remarkable inhibition activity on vesicular monoamine transporter (VMAT2)[1].
[1]. Kilbourn M, et al. Binding of alpha-dihydrotetrabenazine to the vesicular monoamine transporter is stereospecific. Eur J Pharmacol. 1995 May 24;278(3):249-52.
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