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TrkA-IN-3 是一种有效和亚选择性的 TrkA 变构抑制剂,IC50 值为 22.4 nM。TrkA-IN-3 对 TrkA 的选择性超过 TrkB 和 TrkC 8000 倍。TrkA-IN-3 可用于研究疼痛。
TrkA-IN-3 is a potent, subselective and allosteric TrkC. TrkA-IN-3 can be used for the research of pain[1].
TrkA-IN-3 (化合物 5) 在浓度为 1 μM 和 0.1 μM 时对 TrkA 的抑制率分别为 73.9% 和 64.8%[1]。
[1]. Tang S, et, al. Design, development and evaluation of a prodrug-type TrkA-selective inhibitor with antinociceptive effects in vivo. Eur J Med Chem. 2023 Jan 5;245(Pt 2):114901.
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