CARM1-IN-6 (iCARM1) 是一种有效的、选择性的 CARM1 抑制剂, IC50 值为 12.3 μM。CARM1-IN-6 具有抑制细胞生长活性,可用于癌症的研究。
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CARM1-IN-6 (iCARM1) is an effective and selective inhibitor of CARM1 with an IC50 value of 12.3 μM. CARM1-IN-6 exhibits cell growth inhibitory activity and can be used in cancer research[1].
参考文献:
[1]. Peng BL, et al. A CARM1 Inhibitor Potently Suppresses Breast Cancer Both In Vitro and In Vivo. J Med Chem. 2024 May 23;67(10):7921-7934.