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Neratinib (HKI-272)
A dual inhibitor of EGFR and HER2
Mutated EGFR-IN-2
Mutated EGFR-IN-2 (compound 91) 突变选择性的 EGFR 抑制剂,有效抑制单突变体 EGFR (T790M) 和双突变体 EGFR (包括 L858R/T790M (IC50=<1nM) 和 ex19del/T790M),并且可以抑制单一功能获得性突变 EGFR (包括 L858R 和 ex19del) 的活性。Mutated EGFR-IN-2 具有抗肿瘤活性。
LKB1(AAK1 dual inhibitor)
LKB1(AAK1 dual inhibitor) 是一种有效的多激酶抑制剂,对 Pim1/AKK1/MST2/LKB1 的 Kd 值分别为 35 nM/53 nM/75 nM/380 nM,并且还抑制 MPSK1 和 TNIK。
Naquotinib (ASP8273)
An irreversible inhibitor of mutant EGFRs
PIM-1 Inhibitor 2
A potent PIM-1 kinase inhibitor
Avitinib
A selective inhibitor of mutant EGFR
Fludarabine Phosphate (Fludara)
A prodrug form of fludarabine and 2-fluoro-ara-ATP
AZD3759
A brain penetrant inhibitor of EGFR
MM-206
A STAT3 inhibitor
5,15-DPP
NSC 74859
FLLL32
An inhibitor of JAK2/STAT3 signaling
Niclosamide
An anthelmintic mitochondrial uncoupler
STAT5 Inhibitor
Prevents activation of STAT5 via its SH2 domain
NT157
IRS-1/2 抑制剂,抑制 IGF-1R 和 STAT3 信号通路