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Lapatinib
A dual inhibitor of EGFR and ErbB2
Nazartinib mesylate
An inhibitor of mutant EGFR
Neratinib (HKI-272)
A dual inhibitor of EGFR and HER2
Mutated EGFR-IN-2
Mutated EGFR-IN-2 (compound 91) 突变选择性的 EGFR 抑制剂,有效抑制单突变体 EGFR (T790M) 和双突变体 EGFR (包括 L858R/T790M (IC50=<1nM) 和 ex19del/T790M),并且可以抑制单一功能获得性突变 EGFR (包括 L858R 和 ex19del) 的活性。Mutated EGFR-IN-2 具有抗肿瘤活性。
Naquotinib (ASP8273)
An irreversible inhibitor of mutant EGFRs
Avitinib
A selective inhibitor of mutant EGFR
AZD3759
A brain penetrant inhibitor of EGFR
Tyrphostin 9
An inhibitor of EGF receptor kinase
Regorafenib
A multi-kinase inhibitor
WHI-P180 hydrochloride
AV-412 free base
Tesevatinib (XL-647)
Icotinib
An EGFR inhibitor
BGB-283
BGB-283 is a novel and potent Raf Kinase and EGFR inhibitor with IC50 values of 23 and 29 nM for recombinant BRafV600E and EGFR, respectively.
Afatinib(BIBW2992)
A selective dual inhibitor of EGFR/HER2