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MC-Val-Cit-PAB-MMAF是一种偶联药物(drug-linkerconjugateforADC),具有抗肿瘤活性,由抗微管蛋白抑制剂MMAF和组织蛋白酶可降解(cleavable)的linkerMC-Val-Cit-PAB连接而成。
MC-Val-Cit-PAB-MMAF is a drug-linker conjugate for ADC with antitumor activity by using the tubulin inhibitor, MMAF, linked via cathepsin cleavable MC-Val-Cit-PAB.
[1]. Cheng X, et al. MORAb-202, an Antibody-Drug Conjugate Utilizing Humanized Anti-human FRα Farletuzumab and the Microtubule-targeting Agent Eribulin, has Potent Antitumor Activity. Mol Cancer Ther. 2018 Dec;17(12):2665-2675.
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