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AuroraBinhibitor1是一种AuroraB(Aurora-1)抑制剂,Ki值<0.010uM。详细信息请参考专利文献WO2007059299A1中的化合物1-3。
Aurora B inhibitor 1 is an Aurora B (Aurora-1) inhibitor extracted from patent WO2007059299A1, compound 1-3, has a Ki value of <0.010 uM.
Aurora B inhibitor 1 also inhibits JAK3 and JAK2 with Kis of <0.25 μM and <0.10 μM, respectively[1].
[1]. FRAYSSE, Damien, et al. AMINOPYRIMIDINES USEFUL AS KINASE INHIBITORS. WO2007059299A1.
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