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Felcisetrag
Felcisetrag (TD-8954) 是一种具有口服活性,有效和选择性 5-HT4 受体激动剂,具有胃肠道促动力特性。Felcisetrag 对人类重组 5-HT4(c) (h5-HT4(c)) 受体具有高亲和力 (pKi =9.4)。
NLX-204 hydrochloride
NLX-204 is a potent, selective agonist of ERK1/2 phosphorylation-preferring serotonin 5 HT1A receptor with pKi of 10.19.
Hydroxy ziprasidone
Hydroxyziprasidone是Ziprasidone的杂质。Ziprasidone,一种抗精神药物,是5-HT和多巴胺(dopaminereceptor)受体拮抗剂。
Cyclobenzaprine-d3 (hydrochloride) (CRM)
A Certified Reference Material
(±)-CP 55,940-d11
A neuropeptide with diverse biological activities
Keto Ziprasidone
KetoZiprasidone是Ziprasidone的杂质。Ziprasidone,一种抗精神药物,是5-HT和多巴胺(dopaminereceptor)受体拮抗剂。
S 14506
A 5-HT1A receptor agonist
(S)-(-)-Docosahexaenyl-1'-Hydroxy-2'-Propylamide
DHEA的同源物
11C-MK-3168
11C-MK-3168是一种有效的,选择性的,可透过血脑屏障的脂肪酸酰胺水解酶(FAAH)抑制剂,对人,大鼠和恒河猴FAAH的IC50值分别为1.0,1.7和5.5nM。
Sarpogrelate-d3 (hydrochloride)
An internal standard for the quantification of sarpogrelate
Melperone-d4 (hydrochloride)
An internal standard for the quantification of melperone
(S)-(+)-Docosahexaenyl-2'-Hydroxy-1'-Propylamide
4-Ethynyl-L-phenylalanine hydrochloride
4-Ethynyl-L-phenylalanine hydrochloride (4-Ethynyl-L-phenylalanine hydrochloride) 是一种有效的、选择性的、可逆的和竞争性的色氨酸羟化酶 (TPH) 抑制剂,Ki 为 32.6 μM.
Palonosetron N-oxide
A metabolite of palonosetron
Trifluoperazine-d3 (hydrochloride)
An internal standard for the quantification of trifluoperazine