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Indobufen
Indobufen (Ibustrin, K 3920) is a reversible platelet aggregation inhibitor. Indobufen is a reversible inhibitor of platelet cyclooxygenase (Cox) activity and suppresses thromboxane synthesis.
Asaraldehyde
Asarylaldehyde (Asaronaldehyde) 是一种 COX-2 抑制剂,可显着抑制环氧合酶 II (COX-2) 的活性,IC50 值为 100 μg/mL。
Imrecoxib
Imrecoxib(BAP-909)艾瑞昔布是选择性环氧合酶 2 (COX-2) 抑制剂,IC50 值为 18 nM,也可以抑制 COX1 活性,IC50 值为 115 nM。Imrecoxib(BAP-909) 艾瑞昔布具有抗炎作用。
Piroxicam
A COX inhibitor and NSAID
Prostaglandin G2
The first stable intermediate in the COX pathway
N-(4-acetamidophenyl)-Indomethacin amide
Potent and selective reversible inhibitor of COX-2
Acemetacin
An NSAID
Prostaglandin D3
An inhibitor of platelet aggregation
Ginsenoside Rg5
A ginsenoside with diverse biological activities
Polmacoxib
An inhibitor of COX-2 and carbonic anhydrase
Diclofenac Sodium
An NSAID and a COX inhibitor
Rofecoxib
A COX-2 inhibitor
Tryptanthrin
An alkaloid with diverse actions
Tenidap
A COX-1 selective NSAID
Naproxen etemesil (LT-NS 001)
Naproxen etemesil (LT-NS 001) 是一种亲脂性、非酸性、无活性的萘普生前药,一旦被吸收就会水解成具有药理活性的萘普生。