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Lornoxicam
A COX inhibitor and NSAID
Sulindac
A non-selective COX inhibitor
Iguratimod
A DMARD and COX-2 inhibitor
Etoricoxib
A selective COX-2 inhibitor
COX2-IN-1
COX2-IN-1是选择性的,诱导型的COX2抑制剂,IC50值为0.24μM。COX2-IN-1是具有抗炎和止痛活性的抗炎物。
RWJ 63556
RWJ63556是一种可口服的COX-2selective/5-lipoxygenase抑制剂,具有抗炎活性。
Indomethacin
Indomethacin (Indometacin) is a potent, orally active COX1/2 inhibitor with IC50 values of 18 nM and 26 nM for COX-1 and COX-2, respectively.
Nabumetone
An NSAID and a prodrug form of 6-methoxy naphthalene acetic acid
ADDA 5 hydrochloride
ADDA5hydrochloride是一种部分非竞争性的细胞色素c氧化酶(cytochromecoxidase(CcO))抑制剂,可抑制从人胶质瘤细胞和牛心肌细胞中分离纯化的CcO的活性,IC50值分别为18.93μM和31.82μM。
Fenbufen
An NSAID
TFAP
A selective COX-1 inhibitor
NS 398
A selective COX2 inhibitor
(S)-Ketoprofen
A potent inhibitor of COX-1 and COX-2
Bromfenac Sodium
A COX-2 inhibitor
Ampiroxicam
A prodrug of piroxicam