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Bleomycin Sulfate(硫酸博来霉素)
LY 294002
BKT140
A CXCR4 antagonist
Camelliaside A
A flavonoid with radical scavenging and enzyme inhibitory activities
Arginase inhibitor 1
Isopropyl beta-D-thiogalactoside(IPTG)
KP-457
KP‐457?is a selective ADAM17 inhibitor,?which has a reverse-hydroxamate structure. ?ADAM17, also known as TNF-α-converting enzyme, cleaves various molecules such as GPIbα, GPV, and TNF-α.
Betulinic acid
G007-LK
A TNKS1/2 inhibitor
VX-680 (MK-0457,Tozasertib)
KN-92
An inactive control compound for a CaMKII inhibitor
Eflornithine (DFMO)
Eflornithine(DFMO) inhibits polyamine biosynthesis by irreversible inhibition of ornithine decarboxylase(ODC).
D4476
GSK1070916
Elacestrant (RAD1901)
Elacestrant (RAD1901) (RAD1901) 是一种口服选择性雌激素受体降解剂 (SERD),对 ERα 的 IC50 分别为 48 和 870 nM;和ERβ,分别。